CXCR1
CXCR2
CXCR4
CXCR3

CXCR3 選択性拮抗剤

製品コード	製品名	製品説明	Selective / Pan	IC50 / Ki
S8682	AMG 487	AMG 487 is an orally active and selective CXC chemokine receptor 3 (CXCR3) antagonist that inhibits the binding of IP-10 (CXCL10) and ITAC (CXCL11) to CXCR3 with IC50 of 8.0 nM and 8.2 nM, respectively.	Selective	CXCR3-CXCL10, IC50: 8.0 nM; CXCR3-CXCL11, IC50: 8.2 nM