SGK

亜型選択性的な製品

SGK1 SGK2 SGK3

SGK製品

All (3)
SGK阻害剤 (3)
新製品

製品コード	製品名称	製品説明	文献中Selleckの製品使用例	お客様のフィードバック
S7209	GSK650394	GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.	J Clin Invest, 2023, 133(20)e169234 J Leukoc Biol, 2023, qiad025 Reprod Biol Endocrinol, 2023, 21(1):50
S9672	PROTAC SGK3 degrader-1	PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC conjugate of the 308-R SGK inhibitor with the VH032 VHL binding ligand, targeting SGK3 (Serum/Glucocorticoid Regulated Kinase Family Member 3) for degradation.	Front Pharmacol, 2023, 14:1169054 Front Pharmacol, 2023, 14:1169054
S8824	EMD638683	EMD638683 is a highly selective inhibitor of serum- and glucocorticoid-inducible kinase 1 (SGK1) with IC50 of 3 μM. EMD638683 exhibits antihypertensive potency and anti-tumor activity.
S7209	GSK650394	GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively.	J Clin Invest, 2023, 133(20)e169234 J Leukoc Biol, 2023, qiad025 Reprod Biol Endocrinol, 2023, 21(1):50
S9672	PROTAC SGK3 degrader-1	PROTAC SGK3 degrader-1 (SGK3-PROTAC1) is a PROTAC conjugate of the 308-R SGK inhibitor with the VH032 VHL binding ligand, targeting SGK3 (Serum/Glucocorticoid Regulated Kinase Family Member 3) for degradation.	Front Pharmacol, 2023, 14:1169054 Front Pharmacol, 2023, 14:1169054
S8824	EMD638683	EMD638683 is a highly selective inhibitor of serum- and glucocorticoid-inducible kinase 1 (SGK1) with IC50 of 3 μM. EMD638683 exhibits antihypertensive potency and anti-tumor activity.

SGK阻害剤の選択性比較

Tags: SGK inhibitor|SGK agonist|SGK activator|SGK inducer|SGK antagonist|SGK signaling pathway|SGK assay kit