PREP

PREP製品

All (5)
PREP阻害剤 (5)
新製品

製品コード	製品名称	製品説明	文献中Selleckの製品使用例
S2268	Baicalein	Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.	SLAS Discov, 2024, S2472-5552(24)00007-8 Redox Rep, 2023, 28(1):2152607 Microbiol Spectr, 2023, 11(3):e0470222
S2396	Salidroside	Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties.	PLoS One, 2024, 19(7):e0306926 Mol Med Rep, 2023, 27(2)37 Research Square, 2023, 10.21203/rs.3.rs-3696850/v1
S2269	Baicalin	Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.	Ecotoxicol Environ Saf, 2024, 275:116262 Chem Biol Interact, 2024, 387:110820 Int J Mol Sci, 2023, 24(11)9435
S0842	SP-13786	SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S3249	Corypalmine	Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.
S2268	Baicalein	Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor.	SLAS Discov, 2024, S2472-5552(24)00007-8 Redox Rep, 2023, 28(1):2152607 Microbiol Spectr, 2023, 11(3):e0470222
S2396	Salidroside	Salidroside (Rhodioloside), a phenylpropanoid glycoside isolated from Rhodiola rosea, has been reported to have a broad spectrum of pharmacological properties.	PLoS One, 2024, 19(7):e0306926 Mol Med Rep, 2023, 27(2)37 Research Square, 2023, 10.21203/rs.3.rs-3696850/v1
S2269	Baicalin	Baicalin is an inhibitor of prolyl oligopeptidase and also is an allosteric activator of carnitine palmityl transferase 1 (CPT1). Baicalin reduces the expression of NF-κB.	Ecotoxicol Environ Saf, 2024, 275:116262 Chem Biol Interact, 2024, 387:110820 Int J Mol Sci, 2023, 24(11)9435
S0842	SP-13786	SP-13786 (UAMC-1110)(compound 60) is a potent and selective inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP) with IC50 of 3.2 nM and 1.8 μM, respectively.
S3249	Corypalmine	Corypalmine ((R)-(+)-Corypalmine), an alkaloid isolated from Stephania cepharantha, is an inhibitor of prolyl endopeptidase/oligopeptidase (PREP/POP) with IC50 of 128.0 μM.

PREP阻害剤の選択性比較